A fluorescent switchable AIE probe for selective imaging of dipeptidyl peptidase-4 in vitro and in vivo and its application in screening DPP-4 inhibitors.

نویسندگان

  • Yi Wang
  • Xueli Wu
  • Yiyu Cheng
  • Xiaoping Zhao
چکیده

A novel fluorescent probe for in vitro and in vivo imaging of dipeptidyl peptidase-4 (DPP-4) was designed and synthesized. This probe is successfully utilized to screen DPP-4 inhibitors in living 3T3-L1 cells and zebrafish, which provides a novel approach for the discovery of anti-diabetes drugs.

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عنوان ژورنال:
  • Chemical communications

دوره 52 17  شماره 

صفحات  -

تاریخ انتشار 2016